Khavinson BioregulatorTarget: ProstateReproductive

Prostatilen

Samprost · Vitaprost · Сампрост · Простатилен

Prostatilen (Vitaprost/Samprost) is the pharmaceutical prostate extract used in CIS urology. Adjacent to the 41. Libidon is Cytomax; Prostamax is KEDP.

Not FDA-approved - research chemical

Quick answer

What it is: Prostatilen (Vitaprost/Samprost) is the pharmaceutical prostate extract used in CIS urology.

Class and target: Pharmaceutical extract (Cytamin-era) · Prostate

Typical research dose: 5-10 mg rectally or IM

Reconstitution calculator ↓What it is & the evidence on The Bioregulator Atlas →

Research summary, not medical advice.

Reviewed by Kymata Health Editorial Team
Last updated: August 2026Evidence: Low1 peer-reviewed citation
Typical research dose
5-10 mg rectally or IM
Frequency
1× daily for 5-10 days
Half-life
Mixture (variable)
Common vials
5 mg
CAS
N/A (biological extract)
Molecular weight
Mixture (<10 kDa)

Use-case scores

0–10 against the evidence we have, not a gym ranking. Hidden domains do not apply here.

  • Sexual / hormonal3/10

    Russian extract literature. Not a US BPH drug. Not the KEDP tetrapeptide.

Compound card

Class
Bovine prostate polypeptide extract (Cytomax class; not Prostamax KEDP)
Formula
Polypeptide extract (Prostate tissue)
Status
Not FDA-approved · research use
Dose it
5 mg + 1 mL BAC water → 5 mg/mL · 5000 mcg ≈ 100 units (U-100)
Open in calculator

How it works

Prostatilen is a pharmaceutical-grade polypeptide extract derived from the prostate glands of young bulls. Manufactured primarily in Russia and Eastern Europe, it is an injectable therapeutic containing water-soluble peptides with specific tropism (attraction) to the human prostate gland.

It acts by improving prostate microcirculation, reducing tissue edema (swelling), inhibiting leukocyte infiltration (inflammation), and normalizing the secretory function of prostate epithelial cells. It is a widely prescribed clinical treatment in Russia for chronic abacterial prostatitis and benign prostatic hyperplasia (BPH). It works via the same tissue-specific gene regulation pathways as the oral Cytomax version (Libidon), but at a higher, clinical-grade concentration.

Source: PMID: 11713572

Khavinson map

Adjacent (not padded into the 41)
Class
Pharmaceutical extract (Cytamin-era)
Organ
Prostate
Target
Prostate
System
Reproductive
Sequence
Mixture / not a single CAS
Простатилен

Used in bioregulator stacks

Manufacturer-style organ combinations - not FDA protocols. Every name is a live leaf.

The Khavinson school

Prostatilen is filed here as pharmaceutical extract (cytamin-era), targeting the prostate. Khavinson's St. Petersburg group moved from organ extracts (Cytamins) to capsule complexes (Cytomaxes) to synthetic short peptides (Cytogens); most of the evidence comes from that one group, with little independent Western replication.

Read the full background, the proposed epigenetic mechanism, the literature limits, and how we count the canonical 41 on the Khavinson bioregulators index.

History of this molecule

Authorized extract product in its home market, rectal and injectable presentations in labeling folklore. That is a different object than a 10 mg KEDP research vial. We keep the triad honest.

Caveats

Extract. Rising PSA is a workup. Not FDA in the US as this named product for BPH in the American sense.

Full 41-map: Khavinson bioregulators index · Bioregulator stacks

Research Use Cases

  • ✓Chronic abacterial prostatitis
  • ✓Benign prostatic hyperplasia
  • ✓Post-prostatectomy recovery
  • ✓Male genitourinary aging

Dosing

PhaseDoseFrequencyNotes
Clinical Protocol5 - 10 mgDaily IM injection for 5-10 daysRussian clinical standard for prostatitis. Often also available as a rectal suppository (Vitaprost).

Administration

Route / form
Pharmaceutical extract - historically intramuscular or rectal suppository (Prostatilen / Samprost). Not a Cytomax capsule.
Timing
Course-based injectable / extract timing per the pharmaceutical presentation - food does not change an IM or parabulbar shot.
Empty stomach?
No - These are clinic-era injectables or suppositories, not capsules. Food timing does not apply.

Prostatilen: CIS IM extract vs Rectal suppository

CIS IM extract
Bioavailability
CIS pharmaceutical prostate extract (Prostatilen / Vitaprost / Samprost). Documented injectable route is intramuscular. Not KEDP SubQ and not a bladder peptide. Samprost is this extract’s brand, not Chitomur.
Dose note
Ampoule / clinic kit: mix per the pharmaceutical presentation. Do not invent a 5 mg/mL BAC SubQ lifestyle chart for an extract lot. Folklore is 5–10 mg IM daily for 5–10 days. Research-chem “Prostatilen” may be mislabeled KEDP. Match the pharmaceutical presentation.
Advantages
  • Authorized extract product in its home market. Real triad with Libidon and Prostamax.
  • IM is the injectable clinic route, not a 5 mg abdomen lifestyle chart.
  • Food does not change an IM shot.
Considerations
  • Not a US BPH indication. Rising PSA is a workup.
  • Not Vesilut / Chitomur (bladder). Catalogs that file Samprost under bladder are mixing the brand.
  • Identity risk on gray-market powder.
Rectal suppository
Bioavailability
The documented non-injectable presentation is a rectal suppository (Prostatilen / Vitaprost), not a swallowed Libidon Cytomax capsule and not a sublingual tablet. Libidon is the oral prostate complex on a different leaf.
Dose note
Suppository courses follow the home-market insert (order of daily use for several days). If you swallowed a capsule, you bought Libidon or Prostamax cytogen, not this extract.
Advantages
  • Rectal suppository is a real CIS presentation for this extract.
  • Keeps Libidon (Cytomax swallow) separate from the extract.
  • Not a sublingual tablet. Nobody manufactures this SKU that way.
Considerations
  • Suppository ≠ Prostamax KEDP capsule ≠ Libidon capsule.
  • Not tadalafil. Not finasteride.
  • Do not invent a swallowed-extract dose to look complete.
Recommendation: Prostatilen is a CIS prostate extract: IM or rectal suppository. It is not in the 41. It is not Prostamax (KEDP cytogen, capsule-or-vial), not Libidon (prostate Cytomax), not Samprost-as-bladder, and not a 5 mg BAC SubQ chart. Dose the presentation in the box.

Timeline

Day 5-10
Significant subjective reduction in pelvic pain and urinary urgency.
Month 1+
Reduced prostate volume and improved microcirculation.

Who it is for

Chronic Prostatitis / BPH

Moderate

Registered medicine in Russia for acute and chronic prostate inflammation.

Reconstitution

VialWaterConcentrationExample dose
5 mg lyophilized1 mL BAC5 mg/mLExtract kits vs research cakes. Capsules skip the calculator.

Change vial size or water volume? Open the reconstitution calculator.

Safety & Considerations

Registered pharmaceutical in Russia. Clinical trials show very low incidence of systemic side effects. Painful administration (IM injection) compared to oral Libidon.

Regulatory & Legal Status

FDA Status (US)
Research Only
WADA Status (2026)
Not Listed

Not currently on the WADA 2026 Prohibited List. Policies may change - verify before competition.

Classification

Research Chemical

US Compounding: Not eligible / not available

⚠️ This information is for educational purposes only and may not reflect the most current regulatory updates. Always verify with official FDA, WADA, and jurisdiction-specific sources before use.

Limits of current evidence

  • PMID 11713572 is organ-map class, not an FDA BPH program.
  • This site will not treat BPH or prostatitis from this page.

Verdict

Prostatilen is the prostate tissue extract. Prostamax is KEDP. Samprost/Vitaprost are brand collisions. Not finasteride.

Interactions & Contraindications

Standard Cytomax/injection protocol. No significant drug interactions reported in Russian clinical literature.

Synergies & Common Stacks

Prostate extract plus testicular cytogen in Khavinson practice. School pairing, not a male-reproductive NDA on this site.

Prostatilen + Libidon both target prostate health - Prostatilen from natural extract, Libidon from synthetic peptide approach.

Frequently Asked Questions

In the 41?▼
No. Pharma extract layer. Libidon and Prostamax are in the 41.
Vs Prostamax?▼
Mixture extract vs KEDP.
BPH?▼
CIS product history ≠ US BPH indication.
Same as Libidon?▼
Same gland, different class (extract vs Cytomax complex).
Is Samprost a bladder peptide?▼
No. Samprost (Сампрост) is a brand name for this prostate extract (also Vitaprost). The bladder Cytomax is Chitomur; Vesilut is the bladder cytogen. Catalogs that file Samprost under bladder are mixing the brand.
IM, rectal, or capsule?▼
This extract is IM or rectal suppository. Libidon is the swallowed prostate Cytomax. Prostamax is KEDP (capsule-or-vial). Not a sublingual tablet and not a 5 mg BAC abdomen chart.
How does Prostatilen differ from Libidon?▼
They are functionally identical in mechanism. Libidon is classed as a food supplement (Cytomax) for oral preventative use. Prostatilen is a much higher concentration, purified extract classified as a prescription medicine for intramuscular injection to treat acute pathology.
Is Samprost a bladder bioregulator?▼
No. Samprost (Сампрост) is a Russian brand name for the prostate extract also sold as Prostatilen / Vitaprost. The bladder Cytomax is Chitomur; the bladder cytogen is Vesilut. Catalogs that file Samprost under urinary/bladder are mixing up the brand.

References

  1. Khavinson VKh et al. “Tissue-specific effects of peptides.” Bulletin of Experimental Biology and Medicine (2001). PMID: 11713572
Where to get itOral bioregulator

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Prostalon is Vita-Stream's US-made prostate bioregulator (Vita Peptides' own house line), a different product from Prostatilen. No trial has tested it.

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